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Tesofensine

MetabolicMetabolic & Weight LosstherapeuticResearch use only
Educational use only. Not medical advice. Verify all information with primary sources and a licensed clinician before use.
Long; often cited around 9 days for active moieties
Half-life
10
Uses
0.25
Typical
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Overview

Tesofensine is a triple monoamine reuptake inhibitor that blocks the reuptake of serotonin, norepinephrine, and dopamine. Originally developed by NeuroSearch for Parkinson's disease and Alzheimer's disease, it was repurposed for obesity after clinical trial participants experienced significant weight loss. While not technically a peptide, tesofensine is widely discussed in peptide research communities for its potent appetite-suppressing and metabolic effects.

Primary Uses
Weight loss
Appetite reduction
appetite suppression
thermogenesis
energy expenditure enhancement
obesity treatment
Obesity pharmacology
Monoamine reuptake inhibition
Appetite suppression studies
Weight-loss trials
Protocol Reference
Dose
0.25–0.5 mg once daily
Frequency
Once Daily, Morning Preferred
Half-life
Long; often cited around 9 days for active moieties
Route
Oral
Evidence
Phase 2 / Phase 2 clinical trials (disputed)
Research References· 2
Effect of tesofensine on bodyweight loss, body composition, and quality of life in obese patients: a randomised, double-blind, placebo-controlled trial
PubMedPMID 18996750. The Lancet, 2008.
The effect of the triple monoamine reuptake inhibitor tesofensine on energy metabolism and appetite in overweight and moderately obese men
PubMedPMID 20440295. International Journal of Obesity, 2010.
Research Models
Human
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